SCHEMBL299502

SCHEMBL299502

CC(C)(C)OC(=O)N(C(=O)OC(C)(C)C)[C@@H]1C=C[C@H](n2cnc3cnc(Cl)nc32)C1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 3/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
ABCB1 P08183 1/20 0.30
ADCY5 O95622 4/20 0.30
STK17B O94768 1/20 0.30
STK17A Q9UEE5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL239530 0.84 LMNA (0.39) NFKB1NFKB2RELAABCB1ADCY5
SCHEMBL242414 0.78 LMNA (0.38) NFKB1NFKB2RELAABCB1ADCY5
SCHEMBL1401991 0.76 NT5E (0.34) ABCB1ADCY5
SCHEMBL241801 0.75 ADORA3 (0.52)
SCHEMBL4349797 0.74 ADCY5 (0.40) ADCY5
SCHEMBL4349829 0.74 ABCB1 (0.32) ABCB1ADCY5
SCHEMBL4353816 0.74 LMNA (0.37) ABCB1ADCY5
SCHEMBL4432120 0.73 LMNA (0.37) ABCB1ADCY5
SCHEMBL242801 0.73 ADORA1 (0.37)
SCHEMBL1401972 0.72 ADORA1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013211-B1 PURINE DERIVATIVES FOR USE AS ADENOSIN A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2012-03-14 EP disclosed