SCHEMBL29951249

SCHEMBL29951249

COc1ccnc2[nH]cc(C=O)c12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 5/20 0.51
CDK9 P50750 5/20 0.51
CDK5 Q00535 5/20 0.51
CDK5R1 Q15078 5/20 0.51
CCNA2 P20248 4/20 0.51
CDK2 P24941 4/20 0.51
CCNA1 P78396 4/20 0.51
KMT2A Q03164 2/20 0.47
HTR2A P28223 1/20 0.45
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
HASPIN Q8TF76 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SIK1 P57059 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27869093 0.82 KMT2A (0.43) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL29957196 0.80 KMT2A (0.56) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL17843962 0.79 KMT2A (0.51) CCNT1CDK9CDK5KMT2AHTR2A
SCHEMBL1951472 0.78 MAP2K1 (0.50) KMT2AALDH1A1KDM4E
SCHEMBL29954463 0.78 MAP2K1 (0.50) KMT2AALDH1A1KDM4E
SCHEMBL26612367 0.77 MAP3K7 (0.46) KMT2AALDH1A1MAPT
SCHEMBL29956991 0.77 KMT2A (0.36) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL19478523 0.77 CDK2 (0.56) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL20757818 0.76 KMT2A (0.49) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL25249416 0.76 CCNT1 (0.55) CCNT1CDK9CDK5CDK5R1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed