SCHEMBL29952012

SCHEMBL29952012

Nc1ncc(C=O)cc1-c1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.54
FYN P06241 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.47
ERN1 O75460 2/20 0.46
TTK P33981 1/20 0.44
TDO2 P48775 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
PTK2 Q05397 1/20 0.43
MKNK1 Q9BUB5 2/20 0.42
MKNK2 Q9HBH9 2/20 0.42
MEN1 O00255 1/20 0.42
PSIP1 O75475 1/20 0.42
AXL P30530 1/20 0.42
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
CYP19A1 P11511 1/20 0.42
CYP3A4 P08684 4/20 0.42
CYP2A6 P11509 3/20 0.42
CYP2E1 P05181 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29951522 0.84 MAP4K4 (0.51) CHEK2FYNMKNK1AXLMAP4K4
SCHEMBL29951774 0.83 CHEK2 (0.51) CHEK2FYNMKNK1CYP2A6CYP1A2
SCHEMBL2558901 0.78 CHEK2 (0.53) CHEK2FYNMKNK1MAP4K4
SCHEMBL26916929 0.76 CHEK2 (0.55) CHEK2FYNTDO2HSP90AA1HSP90AB1
SCHEMBL29582616 0.76 CHEK2 (0.55) CHEK2FYNTDO2HSP90AA1HSP90AB1
SCHEMBL2561948 0.75 MAP4K4 (0.54) CHEK2FYNTDO2MKNK1MEN1
SCHEMBL3931286 0.75 TTK (0.49) LOXL2ERN1TTKMKNK1MKNK2
SCHEMBL21994688 0.74 PDGFRB (0.61) CHEK2FYNMKNK1MKNK2CYP11B1
SCHEMBL29994102 0.74 PDGFRB (0.61) CHEK2FYNMKNK1MKNK2CYP11B1
SCHEMBL2559978 0.74 ADORA2A (0.49) CYP3A4CYP2C9CYP2C19CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed