SCHEMBL29951774

SCHEMBL29951774

Nc1ncc(C=O)cc1-c1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.51
FYN P06241 2/20 0.49
MAPK1 P28482 2/20 0.41
USP7 Q93009 2/20 0.40
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
AKT1 P31749 1/20 0.38
PIK3CA P42336 1/20 0.38
MET P08581 1/20 0.37
MAP4K4 O95819 4/20 0.37
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
AURKB Q96GD4 1/20 0.36
INCENP Q9NQS7 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP1A2 P05177 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29951522 0.85 MAP4K4 (0.51) CHEK2FYNUSP7MAP4K4MKNK1
SCHEMBL29952012 0.83 CHEK2 (0.54) CHEK2FYNMAP4K4CYP2A6CYP1A2
SCHEMBL2561948 0.82 MAP4K4 (0.54) CHEK2FYNUSP7MAP4K4CYP1A2
SCHEMBL2557950 0.81 MAP4K4 (0.56) CHEK2MAPK1USP7PIK3CAMAP4K4
SCHEMBL2558901 0.75 CHEK2 (0.53) CHEK2FYNUSP7MAP4K4MKNK1
SCHEMBL2554311 0.75 MAP4K4 (0.43) CHEK2FYNMAP4K4KCNH2MINK1
SCHEMBL29582823 0.74 FYN (0.53) CHEK2FYNMAPK1USP7AKT1
SCHEMBL26916746 0.74 FYN (0.53) CHEK2FYNMAPK1USP7AKT1
SCHEMBL2559978 0.72 ADORA2A (0.49) PIK3CDPIK3CGPIK3CAMAP4K4ADORA2A
SCHEMBL29951470 0.71 PIK3CA (0.33) PIK3CAMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed