SCHEMBL299550

SCHEMBL299550

CN1C(=O)CSc2cc(-c3ccc(CC(C#N)NC(=O)C4CCOCC4N)cc3)ccc21

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.57
KCNH2 Q12809 2/20 0.47
CTSK P43235 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299869 0.88 CTSC (0.62) CTSCKCNH2CTSK
SCHEMBL2885832 0.80 CTSC (0.72) CTSCKCNH2CTSK
SCHEMBL2885836 0.80 CTSC (0.72) CTSCKCNH2CTSK
SCHEMBL299257 0.77 CTSC (0.56) CTSCKCNH2CTSK
SCHEMBL299207 0.74 CTSC (0.69) CTSCCTSK
SCHEMBL9886054 0.74 CTSC (0.52) CTSCKCNH2CTSK
SCHEMBL289370 0.73 CTSC (0.72) CTSCCTSK
SCHEMBL25865613 0.73 CTSC (0.64) CTSCKCNH2
SCHEMBL20162065 0.73 CTSC (1.00) CTSCKCNH2
SCHEMBL29433615 0.73 CTSC (1.00) CTSCKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed