SCHEMBL29956409

SCHEMBL29956409

CC(C)(C)OC(=O)N1C(=O)Cc2cc(B(O)O)ccc21

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.40
BCHE P06276 1/20 0.38
NOTUM Q6P988 1/20 0.38
ESR2 Q92731 1/20 0.34
NR1H2 P55055 1/20 0.33
SRD5A1 P18405 1/20 0.32
BUB1 O43683 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
MAPK1 P28482 1/20 0.31
CRBN Q96SW2 2/20 0.31
DDB1 Q16531 1/20 0.31
HDAC1 Q13547 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
NR1I3 Q14994 1/20 0.30
DHODH Q02127 1/20 0.30
DTYMK P23919 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31526050 0.82 PDE5A (0.41) PDE5ABCHENOTUMESR2NR1H2
SCHEMBL17022464 0.82 PDE5A (0.41) PDE5ABCHENOTUMESR2NR1H2
SCHEMBL26647342 0.82 PDE5A (0.41) PDE5ABCHENOTUMESR2SRD5A1
SCHEMBL2673664 0.82 PDE5A (0.41) PDE5ABCHENOTUMESR2MAPT
SCHEMBL2267569 0.81 NOTUM (0.43) PDE5ABCHENOTUMKDM4E
SCHEMBL2419240 0.78 NOTUM (0.62) PDE5ABCHENOTUMKDM4EMAPT
SCHEMBL29541811 0.78 NOTUM (0.62) PDE5ABCHENOTUMKDM4EMAPT
SCHEMBL16830137 0.78 ALDH1A1 (0.47) KDM4EMAPT
SCHEMBL29958326 0.75 GPR119 (0.46) NOTUMESR2NR1H2KDM4EGPR119
SCHEMBL7491697 0.75 GPR119 (0.46) NOTUMESR2NR1H2KDM4EGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed