SCHEMBL29959182

SCHEMBL29959182

CC(C)c1cncc2cnccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
KDM4E B2RXH2 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
HTT P42858 2/20 0.38
ALDH1A1 P00352 1/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
RPS6KA3 P51812 1/20 0.37
IMPDH2 P12268 3/20 0.36
LATS1 O95835 4/20 0.35
LATS2 Q9NRM7 4/20 0.35
HASPIN Q8TF76 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31345172 1.00 LMNA (0.40) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL12045006 1.00 LMNA (0.40) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL12045002 0.86 LMNA (0.39) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL2607319 0.80 LMNA (0.53) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL27317248 0.80 HTT (0.41) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL2607435 0.79 ADRA2A (0.44) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL29875062 0.79 ADRA2A (0.44) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL12789725 0.77 CYP1A2 (0.40) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL20990532 0.77 HASPIN (0.38) LMNAKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL20315030 0.76 RPS6KA3 (0.42) LMNAKDM4ECYP1A2MAPKAPK2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023071998-A1 NOVEL PYRIDO OR TRIAZINE-SUBSTITUTED PYRIDO HETEROCYCLIC COMPOUND 杭州德睿智药科技有限公司 2023-05-04 WO disclosed
CN-115135642-A Inhibitors of mutant forms of EGFR 缆图药品公司 2022-09-30 CN disclosed