SCHEMBL29966580

SCHEMBL29966580

c1ccc(-c2ccc3c(ccc4ncsc43)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.45
RIPK2 O43353 2/20 0.41
EGFR P00533 1/20 0.41
KDR P35968 1/20 0.41
TGFBR1 P36897 1/20 0.41
RIPK3 Q9Y572 1/20 0.41
ESR1 P03372 3/20 0.41
ESR2 Q92731 3/20 0.41
PIK3CA P42336 2/20 0.40
DHFR P00374 1/20 0.40
MAP4K4 O95819 1/20 0.40
PI4KA P42356 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
DYRK1A Q13627 1/20 0.39
GPR84 Q9NQS5 1/20 0.38
TRIM58 Q8NG06 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9196002 1.00 BACE1 (0.45) BACE1RIPK2EGFRKDRTGFBR1
SCHEMBL9191805 0.89 RIPK2 (0.45) BACE1RIPK2EGFRKDRTGFBR1
SCHEMBL29966762 0.86 DYRK1A (0.38) TGFBR1ESR1ESR2PIK3CADYRK1A
SCHEMBL17691815 0.84 ACVR1 (0.39) BACE1RIPK2EGFRKDRTGFBR1
SCHEMBL17691827 0.83 DYRK1A (0.55) BACE1RIPK2EGFRKDRTGFBR1
SCHEMBL29967067 0.81 BACE1 (0.51) BACE1MAP4K4DYRK1ACYP2B6
SCHEMBL29966531 0.79 PGR (0.42) PIK3CADYRK1AALK
SCHEMBL17691991 0.78 RIPK2 (0.36) BACE1RIPK2EGFRKDRTGFBR1
SCHEMBL29871387 0.78 CYP3A4 (0.47) BACE1CYP3A4
SCHEMBL2852558 0.78 CYP3A4 (0.47) BACE1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260122-B Naphthothiazole derivative and synthesis method thereof 陕西科技大学 2024-05-28 CN disclosed
CN-115260122-A Naphthothiazole derivative and synthesis method thereof 陕西科技大学 2022-11-01 CN disclosed