SCHEMBL29966531

SCHEMBL29966531

c1coc(-c2ccc3c(ccc4ncsc43)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.42
ALK Q9UM73 1/20 0.41
CLK4 Q9HAZ1 2/20 0.41
DYRK1A Q13627 1/20 0.41
MCL1 Q07820 8/20 0.41
CCNE2 O96020 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
TOP1 P11387 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
PIM1 P11309 1/20 0.39
HRH1 P35367 2/20 0.37
HRH4 Q9H3N8 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
KCNH2 Q12809 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
ERN1 O75460 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29966580 0.79 BACE1 (0.45) ALKDYRK1APIK3CA
SCHEMBL9196002 0.79 BACE1 (0.45) ALKDYRK1APIK3CA
SCHEMBL29966762 0.74 DYRK1A (0.38) DYRK1APIK3CA
SCHEMBL29967067 0.72 BACE1 (0.51) CLK4DYRK1ACCNE2CCNE1CDK2
SCHEMBL26259745 0.72 PGR (0.62) PGRTOP1PIK3R1PIK3CAPIM1
SCHEMBL29966792 0.70 CYP1A2 (0.43)
SCHEMBL28874637 0.70 BACE1 (0.41) PIM1ERN1
SCHEMBL28874626 0.70 CYP1A2 (0.43)
SCHEMBL9190130 0.70 TYMS (0.40) HRH4
SCHEMBL29966934 0.70 BACE1 (0.41) PIM1ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260122-B Naphthothiazole derivative and synthesis method thereof 陕西科技大学 2024-05-28 CN disclosed
CN-115260122-A Naphthothiazole derivative and synthesis method thereof 陕西科技大学 2022-11-01 CN disclosed