SCHEMBL29967412

SCHEMBL29967412

O=C(O)c1ccn2c(O)c(Cc3ccccc3)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 3/20 0.41
KDM4C Q9H3R0 3/20 0.41
KDM5B Q9UGL1 3/20 0.41
KDM2B Q8NHM5 2/20 0.41
ABCB1 P08183 1/20 0.41
AKT1 P31749 1/20 0.39
AKT2 P31751 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
IP6K1 Q92551 1/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30733946 0.78 PLAU (0.49) ABCB1KDM4EHPGDPTPN1PLAU
SCHEMBL7863078 0.71 KDM4E (0.50) KDM5AKDM4CKDM5BKDM2BKDM4E
SCHEMBL11240930 0.68 KDM4E (0.60) AKT1AKT2KDM4ESMN1; SMN2KMT2A
SCHEMBL17434280 0.68 HDAC1 (0.44) KMT2AMEN1
SCHEMBL1428462 0.67 TDP1 (0.42) AKT1AKT2KDM4ESMN1; SMN2KMT2A
SCHEMBL973778 0.66 TDP1 (0.45) AKT1AKT2KDM4ESMN1; SMN2KMT2A
Diphenylmethane SCHEMBL28928022 0.65 FOLH1 (0.62) LMNAKMT2ATSHR
SCHEMBL28555999 0.65 NPC1 (0.38) AKT1AKT2KMT2AMEN1HTT
SCHEMBL27925527 0.64 KDM4C (0.62) KDM5AKDM4CKDM5BKDM2BKDM4E
SCHEMBL22587714 0.64 NR1H4 (0.43) AKT1AKT2KDM4ELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022188876-A1 FUSED RING HETEROCYCLIC COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AND APPLICATION THEREOF 浙江大学 2022-09-15 WO disclosed