SCHEMBL11240930

SCHEMBL11240930

O=C(O)c1ccn2c(=O)c3ccccc3nc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.60
GLA P06280 3/20 0.60
ALDH1A1 P00352 3/20 0.60
GAA P10253 2/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
HSD17B10 Q99714 3/20 0.52
CASP1 P29466 2/20 0.52
CASP7 P55210 2/20 0.52
AKR1B1 P15121 1/20 0.48
MAPK1 P28482 1/20 0.47
RXFP1 Q9HBX9 2/20 0.45
ATM Q13315 1/20 0.45
AKT1 P31749 1/20 0.44
AKT2 P31751 1/20 0.44
HPGD P15428 3/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
KEAP1 Q14145 1/20 0.43
CYP1B1 Q16678 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28663365 0.82 ALPG (0.48) KDM4EGLAALDH1A1GAASMN1; SMN2
SCHEMBL11759583 0.79 KDM4E (0.64) KDM4EGLAALDH1A1GAASMN1; SMN2
SCHEMBL22059444 0.79 KDM4E (0.64) KDM4EGLAALDH1A1GAASMN1; SMN2
SCHEMBL28679155 0.79 SMN1; SMN2 (0.64) KDM4EGLAALDH1A1GAASMN1; SMN2
SCHEMBL18015436 0.79 KDM4E (0.64) KDM4EGLAALDH1A1GAASMN1; SMN2
SCHEMBL11009983 0.79 PTAFR (0.46) ALPG
SCHEMBL11269027 0.79 ALPG (0.70) KDM4EALDH1A1HSD17B10ATMHPGD
Doqualast SCHEMBL124450 0.78 KDM4E (0.63) KDM4EGLAALDH1A1GAASMN1; SMN2
SCHEMBL11245977 0.78 AKR1B1 (0.71) KDM4EGLAALDH1A1GAASMN1; SMN2
SCHEMBL2427657 0.76 KDM4E (1.00) KDM4EGLAALDH1A1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4332802-A 11-Oxo-11H-pyrido[2,1-b]quinazoline-2-carboxylic acid and salts thereof, antiallergic compositions containing it and methods of suppressing allergic reactions with it BOEHRINGER INGELHEIM KG (DE) 1982-06-01 US disclosed