SCHEMBL29967694

SCHEMBL29967694

C/C(=N\c1cnn(C)c1C(=O)O)N1CCOC[C@H]1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
HIF1A Q16665 1/20 0.33
PRMT5 O14744 2/20 0.32
PIK3CD O00329 2/20 0.32
PIK3R2 O00459 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
PIK3R5 Q8WYR1 1/20 0.32
PIK3R3 Q92569 1/20 0.32
PDCD1 Q15116 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28582531 1.00 VNN1 (0.35) VNN1CA12CA1CA2CA9
SCHEMBL28582530 1.00 VNN1 (0.35) VNN1CA12CA1CA2CA9
SCHEMBL23408498 0.88 CNR2 (0.38) VNN1CA12CA1CA2CA9
SCHEMBL29968500 0.86 CA12 (0.35) VNN1CA12CA1CA2CA9
SCHEMBL23408450 0.77 PIK3CD (0.35) VNN1CA12CA1CA2CA9
SCHEMBL28569870 0.72 ATR (0.34) VNN1ALOX5APFEN1PRMT5
SCHEMBL23629194 0.72 ATR (0.34) VNN1ALOX5APFEN1PRMT5
SCHEMBL24024047 0.71 VNN1 (0.30) VNN1
SCHEMBL23629188 0.70 VNN1 (0.35) VNN1CA12CA1CA2CA9
SCHEMBL28560469 0.70 VNN1 (0.35) VNN1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4063363-A1 PYRAZOLO-HETEROARYL DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF Jiangsu Hengrui Pharmaceuticals Co., Ltd. (CN) 2022-09-28 EP disclosed