SCHEMBL29967798

SCHEMBL29967798

Brc1cccc2[nH]c(-c3ccccc3)nc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 6/20 0.56
PARP1 P09874 3/20 0.56
GAA P10253 6/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
GRIN2B Q13224 1/20 0.50
MGAM O43451 4/20 0.49
SI P14410 4/20 0.49
MGAM2 Q2M2H8 4/20 0.49
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
PTGES O14684 1/20 0.48
RPS6KA3 P51812 1/20 0.46
MAPK13 O15264 1/20 0.46
GCGR P47871 1/20 0.46
MAPK12 P53778 1/20 0.46
MAPK11 Q15759 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5938 1.00 DHODH (0.56) DHODHPARP1GAANPC1RAB9A
SCHEMBL29056629 0.85 GAA (0.68) DHODHPARP1GAANPC1RAB9A
SCHEMBL29056668 0.82 MGAM (0.69) DHODHPARP1GAAMGAMSI
SCHEMBL29056753 0.82 GAA (0.69) PARP1GAAMGAMSIMGAM2
SCHEMBL29056652 0.82 PTGES (0.56) PARP1GAANPC1RAB9AMGAM
SCHEMBL29056720 0.81 PARP1 (0.62) DHODHPARP1GAANPC1RAB9A
SCHEMBL29056651 0.81 MGAM (0.48) DHODHPARP1GAANPC1RAB9A
SCHEMBL29056620 0.81 MGAM (0.51) DHODHPARP1GAAMGAMSI
SCHEMBL3286051 0.81 HDAC6 (0.60) PARP1GAAMGAMSIMGAM2
SCHEMBL31027957 0.80 DHODH (0.59) DHODHPARP1GAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed