SCHEMBL29968017

SCHEMBL29968017

FC(F)(F)Oc1ccnc(Nc2cc(N3CCCC4(CNC4)C3)nc(-c3cccnc3)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF2AK4 Q9P2K8 2/20 0.41
HDAC1 Q13547 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
ABL1 P00519 5/20 0.38
NPY5R Q15761 1/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
GALR2 O43603 2/20 0.36
ROCK1 Q13464 2/20 0.35
CDC42BPB Q9Y5S2 2/20 0.35
ROCK2 O75116 1/20 0.35
CDC42BPA Q5VT25 1/20 0.35
KDM6B O15054 1/20 0.34
NR1I2 O75469 1/20 0.34
CHRNA1 P02708 1/20 0.34
MAOB P27338 1/20 0.34
OPRM1 P35372 1/20 0.34
AHR P35869 1/20 0.34
AVPR1A P37288 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23763325 1.00 EIF2AK4 (0.41) EIF2AK4HDAC1HDAC6ABL1NPY5R
SCHEMBL29969336 0.95 NPY5R (0.37) EIF2AK4HDAC1HDAC6ABL1NPY5R
SCHEMBL23763007 0.95 NPY5R (0.37) EIF2AK4HDAC1HDAC6ABL1NPY5R
Hydrochloric Acid SCHEMBL29967952 0.95 NPY5R (0.37) EIF2AK4HDAC1HDAC6ABL1NPY5R
SCHEMBL29967990 0.92 ALDH1A1 (0.42) ABL1ROCK1CDC42BPBROCK2CDC42BPA
SCHEMBL23763037 0.92 ALDH1A1 (0.42) ABL1ROCK1CDC42BPBROCK2CDC42BPA
Hydrochloric Acid SCHEMBL29968440 0.91 ALDH1A1 (0.41) ABL1ROCK1CDC42BPBROCK2CDC42BPA
SCHEMBL23763045 0.91 MAPKAPK2 (0.38) HDAC1HDAC6ABL1NPY5RROCK1
SCHEMBL29968473 0.91 MAPKAPK2 (0.38) HDAC1HDAC6ABL1NPY5RROCK1
SCHEMBL23763059 0.91 NPY5R (0.38) HDAC1HDAC6ABL1NPY5RGALR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115151534-A Inhibitors of interleukin-1 receptor-related kinase (IRAK)/FMS-like receptor tyrosine kinase (FLT 3), pharmaceutical products thereof, and methods thereof 南京药石科技股份有限公司 2022-10-04 CN claimed
CN-115151534-B Inhibitors of interleukin-1 receptor associated kinase (IRAK)/FMS-like receptor tyrosine kinase (FLT 3), pharmaceutical products thereof and methods of use thereof 南京药石科技股份有限公司 2024-02-06 CN disclosed
CN-115151534-A Inhibitors of interleukin-1 receptor-related kinase (IRAK)/FMS-like receptor tyrosine kinase (FLT 3), pharmaceutical products thereof, and methods thereof 南京药石科技股份有限公司 2022-10-04 CN disclosed