SCHEMBL29972178

SCHEMBL29972178

Cc1cc(N)ccc1Oc1ccncn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.40
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 5/20 0.37
HSP90AA1 P07900 1/20 0.36
MAP4K4 O95819 2/20 0.36
POLB P06746 2/20 0.35
PDE10A Q9Y233 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPT P10636 3/20 0.34
LMNA P02545 1/20 0.34
THRB P10828 1/20 0.34
ALOX15 P16050 1/20 0.34
EGFR P00533 2/20 0.33
RAF1 P04049 1/20 0.33
CASP1 P29466 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 1/20 0.32
GAA P10253 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25383309 0.81 MEN1 (0.45) KDM4EHSP90AA1MAP4K4MEN1KMT2A
SCHEMBL4796549 0.79 KDM4E (0.47) KEAP1ALDH1A1KDM4EMAP4K4POLB
SCHEMBL20605542 0.79 MAP4K4 (0.40) KEAP1ALDH1A1KDM4EMAP4K4POLB
SCHEMBL4797866 0.79 MAP4K4 (0.40) KEAP1ALDH1A1KDM4EHSP90AA1MAP4K4
SCHEMBL12593846 0.79 KEAP1 (0.62) KEAP1ALDH1A1KDM4EMAP4K4POLB
SCHEMBL4799464 0.78 ALOX5AP (0.44) KEAP1ALDH1A1KDM4EMAP4K4POLB
SCHEMBL4796604 0.78 KMT2A (0.49) KEAP1ALDH1A1KDM4EPOLBMEN1
SCHEMBL30354890 0.77 ALDH1A1 (0.42) ALDH1A1KDM4EMAP4K4POLBPDE10A
SCHEMBL9007828 0.77 SMN1; SMN2 (0.56) KEAP1ALDH1A1KDM4EHSP90AA1MAP4K4
SCHEMBL4797567 0.77 ALDH1A1 (0.42) ALDH1A1KDM4EMAP4K4POLBPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107141293-B Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2022-09-23 CN disclosed
CN-115057861-A Nitrogen-containing heterocyclic compound, preparation method, intermediate, composition and application 上海医药集团股份有限公司 2022-09-16 CN disclosed