SCHEMBL29973045

SCHEMBL29973045

COC(=O)c1nn(-c2ccc(C3OCCO3)cn2)cc1F

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 4/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
RAB9A P51151 4/20 0.34
ALDH1A1 P00352 4/20 0.34
PKM P14618 1/20 0.34
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KMT2A Q03164 2/20 0.32
GAA P10253 1/20 0.32
POLB P06746 1/20 0.31
HDAC4 P56524 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27082404 1.00 KDM4E (0.35) KDM4EL3MBTL1NPC1SMN1; SMN2RAB9A
SCHEMBL24409256 0.79 RAB9A (0.32) RAB9AKMT2A
SCHEMBL29972666 0.79 NPC1 (0.36) KDM4ENPC1SMN1; SMN2RAB9AALDH1A1
SCHEMBL24409130 0.79 NPC1 (0.36) KDM4ENPC1SMN1; SMN2RAB9AALDH1A1
SCHEMBL27082391 0.77 MEN1 (0.32) KMT2A
SCHEMBL29972876 0.77 MEN1 (0.32) KMT2A
SCHEMBL27082322 0.76 CYP11B1 (0.31)
SCHEMBL29972943 0.76 CYP11B1 (0.31)
SCHEMBL24955122 0.72 MAPK1 (0.53) KDM4EL3MBTL1NPC1SMN1; SMN2RAB9A
SCHEMBL20176923 0.70 EGLN1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022199503-A1 USE OF HETEROCYCLIC COMPOUND IN TREATING DISEASES RELATED TO KINASE DRUG-RESISTANT MUTATION AND METHOD THEREFOR 四川科伦博泰生物医药股份有限公司 2022-09-29 WO disclosed