SCHEMBL29976161

SCHEMBL29976161

OCc1ccc(N2CC3(CC3)C2)nc1Cl

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
HPGD P15428 3/20 0.32
HSD17B10 Q99714 3/20 0.32
TSHR P16473 2/20 0.32
HIF1A Q16665 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP1A2 P05177 1/20 0.32
SORD Q00796 2/20 0.32
NR1I2 O75469 1/20 0.31
HSD11B1 P28845 1/20 0.31
USP2 O75604 1/20 0.31
KLKB1 P03952 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ADRB2 P07550 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23753976 1.00 ALDH1A1 (0.32) ALDH1A1HPGDHSD17B10TSHRHIF1A
SCHEMBL31033204 0.81 KLKB1 (0.40) ALDH1A1HPGDHSD17B10TSHRHIF1A
SCHEMBL21712931 0.81 KLKB1 (0.40) ALDH1A1HPGDHSD17B10TSHRHIF1A
SCHEMBL23769138 0.81 ALDH1A1 (0.32) ALDH1A1HPGDHSD17B10TSHRHIF1A
SCHEMBL23754040 0.79 TRPV3 (0.34) ALDH1A1HPGDHSD17B10TSHRHIF1A
SCHEMBL31357730 0.79 TRPV3 (0.34) ALDH1A1HPGDHSD17B10TSHRHIF1A
SCHEMBL23769144 0.75 SMPD3 (0.38) SORDKLKB1
SCHEMBL12993437 0.75 GAA (0.46) ALDH1A1TSHRCYP2D6CYP1A2USP2
SCHEMBL23753979 0.75 KLKB1 (0.34) KLKB1ADRB2
SCHEMBL31357699 0.75 KLKB1 (0.34) KLKB1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115087652-B Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2024-05-07 CN disclosed
CN-115087652-A Heteroaromatic carboxamide derivatives as plasma kallikrein inhibitors 勃林格殷格翰国际有限公司 2022-09-20 CN disclosed