SCHEMBL29977356

SCHEMBL29977356

C#Cc1cccc2cc(N)ccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.53
ALDH1A1 P00352 6/20 0.43
HSD17B10 Q99714 4/20 0.43
CYP3A4 P08684 3/20 0.43
CASP1 P29466 4/20 0.42
ALOX15 P16050 2/20 0.42
CASP7 P55210 2/20 0.42
HBB P68871 1/20 0.42
HIF1A Q16665 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.40
MAPT P10636 4/20 0.36
KDM4E B2RXH2 3/20 0.36
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 2/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
TSHR P16473 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL689485 1.00 PLAU (0.53) PLAUALDH1A1HSD17B10CYP3A4CASP1
SCHEMBL28989115 0.90 PLAU (0.45) PLAUALDH1A1HSD17B10CYP3A4CASP1
SCHEMBL688709 0.85 CTDSP1 (0.53) PLAUALDH1A1HSD17B10CYP3A4CASP1
SCHEMBL29061925 0.82 CTDSP1 (0.41) PLAUALDH1A1HSD17B10CYP3A4CASP1
SCHEMBL9097608 0.81 PLAU (0.53) PLAUALDH1A1HSD17B10CYP3A4CASP1
SCHEMBL11718995 0.81 PLAU (0.53) PLAUALDH1A1HSD17B10CYP3A4CASP1
SCHEMBL5438141 0.79 CYP1B1 (0.41) PLAUALDH1A1HSD17B10CASP1HIF1A
SCHEMBL689900 0.78 ALDH1A1 (0.40) PLAUALDH1A1HSD17B10CYP3A4CASP1
SCHEMBL30579742 0.78 CYP1A1 (0.32) PLAUCYP1A1CYP1B1
SCHEMBL9928987 0.77 CYP1B1 (0.40) ALDH1A1HSD17B10HIF1AKDM4ECYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026101924-A1 KRAS MODULATORS ALTEROME THERAPEUTICS, INC. (US) 2026-05-15 WO disclosed
US-12528828-B2 Substituted pyrido[4,3-d]pyrimidines as KRAS modulators ALTEROME THERAPEUTICS, INC. (US) 2026-01-20 US disclosed
US-20250346610-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS ALTEROME THERAPEUTICS INC (US) 2025-11-13 US disclosed
US-12466842-B2 Substituted pyrido [4,3-d]pyrimidines as KRAS modulators ALTEROME THERAPEUTICS, INC. (US) 2025-11-11 US disclosed
US-20250282799-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS ALTEROME THERAPEUTICS, INC. 2025-09-11 US disclosed
US-20250186456-A1 PYRIMIDINE-FUSED CYCLIC COMPOUND AND PREPARATION METHOD AND USE THEREOF GENFLEET THERAPEUTICS (SHANGHAI) INC. (CN) 2025-06-12 US disclosed
US-20250179093-A1 KRAS MODULATORS ALTEROME THERAPEUTICS, INC. 2025-06-05 US disclosed
WO-2025059040-A1 MUTANT KRAS MODULATORS AND USES THEREOF NEWAVE PHARMACEUTICAL INC. (US) 2025-03-20 WO disclosed
EP-4397664-A1 PYRIMIDINE-FUSED CYCLIC COMPOUND AND PREPARATION METHOD AND USE THEREOF Genfleet Therapeutics (Shanghai) Inc. (CN) 2024-07-10 EP disclosed
CN-117222650-A Pyridine or pyrimido-ring compound, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2023-12-12 CN disclosed
WO-2022228568-A1 PYRIDINO- OR PYRIMIDO-CYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 劲方医药科技(上海)有限公司 2022-11-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250179093-A1 KRAS MODULATORS KRAS, NRAS, HRAS PLAU 3466/4885ALDH1A1 4071/4885HSD17B10 3898/4885
US-20250346610-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS KRAS, NRAS, HRAS PLAU 3213/4885ALDH1A1 3593/4885HSD17B10 4743/4885
US-12466842-B2 Substituted pyrido [4,3-d]pyrimidines as KRAS modulators KRAS, NRAS, HRAS PLAU 3213/4885ALDH1A1 3593/4885HSD17B10 4743/4885
US-20250186456-A1 PYRIMIDINE-FUSED CYCLIC COMPOUND AND PREPARATION METHOD AND USE THEREOF KRAS, NRAS, TP53 PLAU 3711/4885ALDH1A1 3323/4885HSD17B10 3915/4885
US-20250282799-A1 SUBSTITUTED PYRIDO[4,3-d]PYRIMIDINES AS KRAS MODULATORS KRAS, NRAS, HRAS PLAU 3213/4885ALDH1A1 3593/4885HSD17B10 4743/4885
US-12528828-B2 Substituted pyrido[4,3-d]pyrimidines as KRAS modulators KRAS, NRAS, HRAS PLAU 4517/4885ALDH1A1 1854/4885HSD17B10 2486/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.