SCHEMBL29977360

SCHEMBL29977360

c1ccc2c3c(cnc2c1)NCN3

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
GPR3 P46089 1/20 0.42
NCF1 P14598 2/20 0.37
CYP1A2 P05177 2/20 0.36
ADRB2 P07550 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.35
PDPK1 O15530 1/20 0.35
CA12 O43570 1/20 0.35
PARP1 P09874 1/20 0.35
ALOX15 P16050 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CA9 Q16790 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
ERN1 O75460 1/20 0.35
TOP2A P11388 1/20 0.35
MAPT P10636 1/20 0.34
NISCH Q9Y2I1 1/20 0.34
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33
PI4K2A Q9BTU6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15064194 1.00 KDM4E (0.42) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL25666734 0.85 KDM4E (0.42) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL1859512 0.77 KDM4E (0.43) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL25666728 0.74 KDM4E (0.39) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL25666751 0.74 KDM4E (0.39) KDM4EGPR3NCF1ADRB2LOXL2
SCHEMBL11880018 0.74 KDM4E (0.36) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL12406712 0.72 KDM4E (0.44) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL1770055 0.69 KDM4E (0.41) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL30972078 0.68 GPR3 (0.48) KDM4EGPR3NCF1CYP1A2ADRB2
SCHEMBL11258247 0.68 GPR3 (0.40) KDM4EGPR3NCF1LOXL2PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022161420-A1 CLASS OF HETEROAROMATIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海翊石医药科技有限公司 2022-08-04 WO disclosed