SCHEMBL25666751

SCHEMBL25666751

c1ccc2c3c(cnc2c1)CNCN3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.39
GPR3 P46089 1/20 0.39
NCF1 P14598 2/20 0.36
ADRB2 P07550 1/20 0.36
HRH4 Q9H3N8 1/20 0.33
TOP2A P11388 1/20 0.33
ERN1 O75460 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
PDPK1 O15530 1/20 0.33
CA12 O43570 1/20 0.33
PARP1 P09874 1/20 0.33
ALOX15 P16050 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CA9 Q16790 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
HTR2C P28335 1/20 0.32
SSTR1 P30872 1/20 0.32
SSTR2 P30874 1/20 0.32
SSTR4 P31391 1/20 0.32
SSTR3 P32745 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12406712 0.86 KDM4E (0.44) KDM4EGPR3NCF1ADRB2HRH4
SCHEMBL25666746 0.79 LMNA (0.41) KDM4EMAPT
SCHEMBL1770055 0.76 KDM4E (0.41) KDM4EGPR3NCF1ADRB2TOP2A
SCHEMBL4910013 0.76 GPR3 (0.41) KDM4EGPR3NCF1ADRB2HRH4
SCHEMBL31503196 0.74 KDM4E (0.42) KDM4EGPR3NCF1ADRB2HRH4
SCHEMBL15064194 0.74 KDM4E (0.42) KDM4EGPR3NCF1ADRB2TOP2A
SCHEMBL29977360 0.74 KDM4E (0.42) KDM4EGPR3NCF1ADRB2TOP2A
SCHEMBL25666733 0.73 KDM4E (0.39) KDM4EGPR3NCF1ADRB2HTR2C
SCHEMBL25666728 0.73 KDM4E (0.39) KDM4EGPR3NCF1ADRB2TOP2A
SCHEMBL25666747 0.72 KDM4E (0.38) KDM4EGPR3NCF1ADRB2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109909-A1 AROMATIC HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND USES THEREOF 上海翊石医药科技有限公司 2023-06-22 WO disclosed