SCHEMBL29977658

SCHEMBL29977658

CCOC(=O)c1cnc(Nc2ccc3c(=O)ccn(C)c3c2)s1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.45
AURKB Q96GD4 1/20 0.45
P2RX3 P56373 4/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MAPT P10636 4/20 0.41
NPC1 O15118 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
DHODH Q02127 7/20 0.40
CDC7 O00311 1/20 0.39
DBF4 Q9UBU7 1/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034834 0.77 MAPT (0.54) AURKAAURKBRAB9ASMN1; SMN2MAPT
SCHEMBL5035841 0.76 MAPK13 (0.56) P2RX3RAB9ASMN1; SMN2MAPTNPC1
SCHEMBL23334316 0.72 DHODH (0.56) AURKAAURKBP2RX3RAB9ASMN1; SMN2
SCHEMBL10235581 0.71 DHODH (0.58) AURKAAURKBRAB9ASMN1; SMN2MAPT
SCHEMBL29976800 0.69 SMN1; SMN2 (0.36) RAB9ASMN1; SMN2NPC1HPGDDHODH
SCHEMBL29976542 0.68 SMN1; SMN2 (0.41) RAB9ASMN1; SMN2NPC1HPGDKMT2A
SCHEMBL29977188 0.68 SMN1; SMN2 (0.40) P2RX3RAB9ASMN1; SMN2NPC1HPGD
SCHEMBL29976559 0.68 SMN1; SMN2 (0.50) RAB9ASMN1; SMN2NPC1HPGDDHODH
SCHEMBL12291072 0.68 CDC7 (0.55) AURKAAURKBRAB9ASMN1; SMN2MAPT
SCHEMBL525917 0.68 RAB9A (0.50) RAB9ASMN1; SMN2MAPTNPC1CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115403558-A Aromatic heterocyclic compound with antitumor activity and preparation method and application thereof 河南真实生物科技有限公司 2022-11-29 CN disclosed