SCHEMBL29978285

SCHEMBL29978285

O=C(CN1CCc2sc(-c3noc(C(F)(F)F)n3)cc2C1)Nc1cncnc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 8/20 0.40
HDAC6 Q9UBN7 8/20 0.38
HDAC1 Q13547 6/20 0.38
HDAC8 Q9BY41 6/20 0.38
HDAC5 Q9UQL6 4/20 0.36
HDAC3 O15379 3/20 0.36
HDAC7 Q8WUI4 3/20 0.36
HDAC2 Q92769 3/20 0.36
HDAC9 Q9UKV0 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
DRD2 P14416 2/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
DRD4 P21917 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978357 0.90 HDAC4 (0.49) HDAC4HDAC6HDAC1HDAC8DRD2
SCHEMBL29978125 0.90 KMT2A (0.48) HDAC4MEN1KMT2AALDH1A1NPSR1
SCHEMBL29978399 0.89 HDAC4 (0.45) HDAC4HDAC6HDAC1HDAC8HDAC5
SCHEMBL29978367 0.88 SMN1; SMN2 (0.43) HDAC4HDAC6HDAC1HDAC8HDAC5
SCHEMBL29977954 0.88 KMT2A (0.47) HDAC4HDAC6HDAC1HDAC8HDAC5
SCHEMBL29978433 0.88 HDAC4 (0.41) HDAC4HDAC6HDAC1HDAC8HDAC5
SCHEMBL29978116 0.88 HDAC4 (0.38) HDAC4HDAC6HDAC1HDAC8HDAC5
SCHEMBL29978122 0.86 PRMT5 (0.44) HDAC4HDAC6HDAC1ALDH1A1KDM4E
SCHEMBL29978163 0.86 PRMT5 (0.44) HDAC4HDAC6HDAC1HDAC8MEN1
SCHEMBL29977951 0.86 MAPT (0.40) HDAC4HDAC6HDAC1HDAC8HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed