SCHEMBL29978522

SCHEMBL29978522

O=C(c1ccc(F)cc1F)N1CCc2cc(-c3noc(C(F)(F)F)n3)sc2C1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HDAC6 Q9UBN7 10/20 0.41
HDAC4 P56524 8/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC1 Q13547 3/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978177 0.93 MEN1 (0.41) MEN1KMT2AHDAC6HDAC4HDAC8
SCHEMBL29978728 0.90 HDAC6 (0.44) MEN1KMT2AHDAC6HDAC4HDAC8
SCHEMBL29978604 0.89 HDAC4 (0.50) HDAC6HDAC4HDAC8HDAC2HDAC1
SCHEMBL29977903 0.85 TAS1R3 (0.43) MEN1KMT2AHDAC6HDAC4HDAC8
SCHEMBL29977911 0.85 HDAC4 (0.44) HDAC6HDAC4HDAC8HDAC2HDAC1
SCHEMBL29978949 0.85 HDAC4 (0.41) HDAC6HDAC4HDAC8HDAC2HDAC1
SCHEMBL29978213 0.84 HDAC4 (0.50) HDAC6HDAC4HDAC8HDAC2HDAC1
SCHEMBL29978646 0.84 HDAC4 (0.48) MEN1KMT2AHDAC6HDAC4HDAC8
SCHEMBL29978650 0.84 HDAC4 (0.48) MEN1KMT2AHDAC6HDAC4HDAC8
SCHEMBL29977922 0.84 ALDH1A1 (0.47) HDAC6HDAC4HDAC8HDAC2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed