SCHEMBL29979225

SCHEMBL29979225

OCc1ccnc(-c2ccc(N3CCOCC3)c(F)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
PIK3CA P42336 2/20 0.46
PIK3CD O00329 1/20 0.46
PDE3B Q13370 4/20 0.45
PDE3A Q14432 4/20 0.45
HTT P42858 1/20 0.45
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
RAB9A P51151 1/20 0.44
JAK2 O60674 1/20 0.44
JAK3 P52333 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MTOR P42345 3/20 0.43
PIK3CG P48736 1/20 0.43
AOC3 Q16853 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29979627 0.81 TLR9 (0.50) NPC1PIK3CAPIK3CDTSHRJAK2
SCHEMBL28475576 0.81 TLR9 (0.50) NPC1PIK3CAPIK3CDTSHRJAK2
SCHEMBL28899916 0.78 PIK3CA (0.56) PIK3CAPIK3CDJAK2MTORPIK3CG
SCHEMBL29979620 0.78 PIK3CA (0.56) PIK3CAPIK3CDJAK2MTORPIK3CG
SCHEMBL29979116 0.77 CNR2 (0.51) PIK3CAPIK3CDHPGDALOX15ALDH1A1
SCHEMBL22262619 0.73 HRH3 (0.56) NPC1PIK3CAPIK3CDHTTHPGD
SCHEMBL20745974 0.72 HRH3 (0.55) NPC1PIK3CAPIK3CDHPGDSMN1; SMN2
SCHEMBL20745049 0.71 PIK3CA (0.49) PIK3CAPIK3CDHTTHPGDALDH1A1
SCHEMBL22262379 0.71 KDM4E (0.47) PIK3CAPIK3CDHPGDALDH1A1LMNA
SCHEMBL15349904 0.70 IDO1 (0.45) NPC1MAPK1RAB9ASYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022216945-A1 MACROCYCLIC MCL1 INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-10-13 WO disclosed