SCHEMBL29979620

SCHEMBL29979620

OCc1ccnc(-c2cccc(N3CCOCC3)c2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.56
PIK3CD O00329 3/20 0.56
MTOR P42345 4/20 0.47
PIK3CG P48736 1/20 0.47
CAMK2D Q13557 1/20 0.47
PLOD2 O00469 2/20 0.46
PLOD3 O60568 2/20 0.46
PLOD1 Q02809 2/20 0.46
KDM1A O60341 1/20 0.46
HDAC1 Q13547 1/20 0.46
KMO O15229 1/20 0.46
TLR9 Q9NR96 1/20 0.45
RPS6KA3 P51812 1/20 0.44
AGXT P21549 1/20 0.44
CFTR P13569 1/20 0.43
JMJD6 Q6NYC1 1/20 0.43
JAK2 O60674 1/20 0.43
MAPK8 P45983 1/20 0.43
MAPK10 P53779 1/20 0.43
DHFR P00374 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28899916 1.00 PIK3CA (0.56) PIK3CAPIK3CDMTORPIK3CGCAMK2D
SCHEMBL28475576 0.85 TLR9 (0.50) PIK3CAPIK3CDMTORPIK3CGHDAC1
SCHEMBL29979627 0.85 TLR9 (0.50) PIK3CAPIK3CDMTORPIK3CGHDAC1
SCHEMBL14961828 0.82 DHFR (0.54) PIK3CAPIK3CDMTORPIK3CGCAMK2D
SCHEMBL20745049 0.81 PIK3CA (0.49) PIK3CAPIK3CDMTORPIK3CG
SCHEMBL20745473 0.79 ABL1 (0.50) PIK3CAPIK3CDMTORPIK3CG
SCHEMBL29979225 0.78 NPC1 (0.46) PIK3CAPIK3CDMTORPIK3CGJAK2
SCHEMBL20745060 0.78 ALDH1A1 (0.53)
SCHEMBL10885415 0.77 CDK1 (0.45) PIK3CAPIK3CDPIK3CGPLOD2PLOD3
SCHEMBL29380102 0.77 CDK1 (0.45) PIK3CAPIK3CDPIK3CGPLOD2PLOD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022216945-A1 MACROCYCLIC MCL1 INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-10-13 WO disclosed