SCHEMBL29979116

SCHEMBL29979116

OCc1ccnc(-c2ccc(N3CCOCC3)nc2)n1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 8/20 0.51
PIK3CD O00329 2/20 0.48
PIK3CA P42336 2/20 0.48
ALDH1A1 P00352 2/20 0.47
ATR Q13535 1/20 0.45
ATRIP Q8WXE1 1/20 0.45
AOC3 Q16853 2/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ERN1 O75460 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978664 0.86 ALDH1A1 (0.52) ALDH1A1ALOX15HSD17B10
SCHEMBL29979627 0.84 TLR9 (0.50) PIK3CDPIK3CAAOC3KDM4E
SCHEMBL28475576 0.84 TLR9 (0.50) PIK3CDPIK3CAAOC3KDM4E
SCHEMBL25082177 0.82 CNR2 (0.52) CNR2PIK3CDPIK3CAALDH1A1AOC3
SCHEMBL29979225 0.77 NPC1 (0.46) PIK3CDPIK3CAALDH1A1AOC3HPGD
SCHEMBL29979620 0.76 PIK3CA (0.56) PIK3CDPIK3CA
SCHEMBL28899916 0.76 PIK3CA (0.56) PIK3CDPIK3CA
SCHEMBL22262619 0.75 HRH3 (0.56) PIK3CDPIK3CAALDH1A1KDM4EHPGD
SCHEMBL1310183 0.75 PIK3CA (0.72) CNR2PIK3CDPIK3CAALDH1A1
SCHEMBL20745974 0.74 HRH3 (0.55) PIK3CDPIK3CAALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022216945-A1 MACROCYCLIC MCL1 INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-10-13 WO disclosed