SCHEMBL29980240

SCHEMBL29980240

FC(F)(F)c1c(Br)ccc2[nH]ncc12

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.50
AXL P30530 2/20 0.50
TRPA1 O75762 2/20 0.44
PTPN6 P29350 1/20 0.40
METAP2 P50579 5/20 0.39
CSNK2A1 P68400 1/20 0.38
IDO1 P14902 3/20 0.37
TDO2 P48775 3/20 0.37
CDK2 P24941 4/20 0.36
CCNA1 P78396 4/20 0.36
FLT3 P36888 3/20 0.36
PBK Q96KB5 1/20 0.36
CYP1A2 P05177 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28799165 1.00 NOS1 (0.50) NOS1AXLTRPA1PTPN6METAP2
SCHEMBL25367669 0.80 AXL (0.51) NOS1AXLTRPA1METAP2IDO1
SCHEMBL18456308 0.79 AXL (0.50) NOS1AXLTRPA1METAP2IDO1
SCHEMBL5404571 0.79 AXL (0.50) NOS1AXLTRPA1METAP2IDO1
SCHEMBL767674 0.76 NOS1 (0.55) NOS1AXLTRPA1PTPN6METAP2
SCHEMBL29383280 0.75 AXL (0.59) NOS1AXLTRPA1PTPN6METAP2
SCHEMBL19617855 0.75 AXL (0.59) NOS1AXLTRPA1PTPN6METAP2
SCHEMBL2427200 0.75 AXL (0.46) AXLTRPA1METAP2CDK2CCNA1
SCHEMBL5417197 0.75 METAP2 (0.47) AXLTRPA1METAP2IDO1FLT3
SCHEMBL12293667 0.75 AXL (0.46) NOS1AXLTRPA1METAP2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212819-A1 INDAZOLE DERIVATIVES AS ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2022-10-06 WO disclosed