SCHEMBL29980428

SCHEMBL29980428

C[Si](C)(C)C#Cc1cc(Cl)cc([N+](=O)[O-])c1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.41
ALDH1A1 P00352 4/20 0.40
TDP1 Q9NUW8 1/20 0.40
TSHR P16473 2/20 0.36
S1PR4 O95977 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8490064 1.00 VCAM1 (0.41) VCAM1ALDH1A1TDP1TSHRS1PR4
SCHEMBL27088355 0.81 VCAM1 (0.41) VCAM1TSHR
SCHEMBL29979560 0.81 VCAM1 (0.41) VCAM1TSHR
SCHEMBL852832 0.78 TSHR (0.38) TSHR
SCHEMBL30956694 0.77 ALDH1A1 (0.46) VCAM1ALDH1A1
SCHEMBL529557 0.77 VCAM1 (0.39) VCAM1ALDH1A1TSHR
SCHEMBL27198413 0.75 VCAM1 (0.42) VCAM1ALDH1A1TDP1TSHR
SCHEMBL1477526 0.75 ALDH1A1 (0.52) ALDH1A1TDP1TSHR
SCHEMBL3771130 0.74 VCAM1 (0.74) VCAM1ALDH1A1TDP1TSHR
SCHEMBL16956247 0.74 VCAM1 (0.47) VCAM1ALDH1A1TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4320109-A1 HETEROCYCLIC DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE TREATMENT OR AMELIORATION OF CANCER Tolremo Therapeutics AG (CH) 2024-02-14 EP disclosed
WO-2022214606-A1 HETEROCYCLIC DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE TREATMENT OR AMELIORATION OF CANCER TOLREMO THERAPEUTICS AG (CH) 2022-10-13 WO disclosed