SCHEMBL29993754

SCHEMBL29993754

NC(=O)c1nc2ccccc2cc1C(C=O)Cc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MAPT P10636 3/20 0.38
IKBKB O14920 2/20 0.36
GRM2 Q14416 3/20 0.36
LMNA P02545 2/20 0.36
POLB P06746 1/20 0.36
STAT3 P40763 1/20 0.36
ALOX5 P09917 1/20 0.36
EGFR P00533 1/20 0.36
TOP2A P11388 1/20 0.36
TOP2B Q02880 1/20 0.36
IDO1 P14902 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SCN9A Q15858 2/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30412340 0.91 ALDH1A1 (0.40) SMN1; SMN2MAPTIKBKBKDM4EALDH1A1
SCHEMBL30411703 0.89 PIN1 (0.36) HTTSMN1; SMN2MAPTIKBKBGRM2
SCHEMBL29994547 0.89 SLC1A1 (0.39) IKBKBALOX5PIN1
SCHEMBL29994296 0.84 ALDH1A1 (0.37) SMN1; SMN2MAPTIKBKBLMNAKDM4E
SCHEMBL30412565 0.79 IKBKB (0.40) HTTMAPTIKBKBLMNAPOLB
SCHEMBL29994393 0.74 BACE1 (0.41) SMN1; SMN2IKBKBLMNAALOX5KDM4E
SCHEMBL30412369 0.72 ALDH1A1 (0.40) SMN1; SMN2MAPTKDM4EALDH1A1MEN1
SCHEMBL28172319 0.70 IKBKB (0.49) SMN1; SMN2MAPTIKBKBSTAT3KDM4E
SCHEMBL4945097 0.70 HTT (0.42) HTTSMN1; SMN2MAPTIKBKBGRM2
SCHEMBL31674405 0.68 IKBKB (0.53) SMN1; SMN2MAPTIKBKBGRM2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4098258-A1 PHARMACEUTICAL USE OF KETOAMIDE-BASED COMPOUND Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2022-12-07 EP claimed
CN-113197895-B Pharmaceutical application of ketoamide compound 中国科学院上海药物研究所 2023-06-20 CN disclosed
EP-4098258-A1 PHARMACEUTICAL USE OF KETOAMIDE-BASED COMPOUND Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2022-12-07 EP disclosed