SCHEMBL29997803

SCHEMBL29997803

COC(=O)c1cc(O)c(C(=O)OC)s1.COC(=O)c1sc(C(=O)OC)c([N+](=O)[O-])c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COMT P21964 8/20 0.50
MAPT P10636 2/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
USP10 Q14694 1/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
NFKB1 P19838 1/20 0.34
XDH P47989 1/20 0.34
GFER P55789 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
FUT7 Q11130 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
OPRD1 P41143 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1846609 0.86 COMT (0.51) COMTMAPTHTTSMN1; SMN2MEN1
SCHEMBL577650 0.81 MAPT (0.45) MAPTSMN1; SMN2KMT2AKDM4ELMNA
SCHEMBL3231061 0.74 USP10 (0.48) COMTMAPTMEN1KMT2AUSP10
SCHEMBL2978000 0.74 COMT (0.49) COMTMAPTHTTSMN1; SMN2MEN1
SCHEMBL577651 0.73 MAPT (0.44) MAPTMEN1KMT2AKDM4ELMNA
SCHEMBL29997056 0.73 OPRD1 (0.39) MAPTSMN1; SMN2KMT2AKDM4ELMNA
SCHEMBL1561317 0.72 OPRD1 (0.43) MAPTSMN1; SMN2KDM4ELMNAPOLB
SCHEMBL17203079 0.70 GSK3B (0.52) MAPTHTTSMN1; SMN2MEN1KMT2A
SCHEMBL1844332 0.69 SMN1; SMN2 (0.57) COMTMAPTHTTSMN1; SMN2MEN1
SCHEMBL23459705 0.68 COMT (0.52) COMTMAPTHTTSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4069369-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME Schrödinger, Inc. (US) 2022-10-12 EP disclosed