SCHEMBL23459705

SCHEMBL23459705

COC(=O)c1scc(O)c1[N+](=O)[O-]

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
COMT P21964 7/20 0.52
SMN1; SMN2 Q16637 1/20 0.44
ALDH1A1 P00352 3/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 1/20 0.38
SLC10A6 Q3KNW5 1/20 0.38
POLB P06746 2/20 0.38
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28866506 0.83 COMT (0.46) COMTSMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL23485294 0.82 SMN1; SMN2 (0.46) COMTSMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL23485282 0.79 GPR35 (0.36) COMTALDH1A1
SCHEMBL6303498 0.77 KDM4E (0.38) COMTSMN1; SMN2KDM4EPOLB
SCHEMBL23485684 0.75 COMT (0.40) COMTSMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL9442593 0.74 KDM4E (0.45) COMTSMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL13545969 0.73 ALDH1A1 (0.49) COMTSMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL24210733 0.73 MAPT (0.43) SMN1; SMN2MAPTKDM4EPOLB
SCHEMBL1846609 0.72 COMT (0.51) COMTSMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL28290128 0.72 ALDH1A1 (0.48) COMTALDH1A1MAPTKDM4ESLC10A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. 2023-11-16 US disclosed
CN-116490507-A Heterocyclic condensation CDC7 kinase inhibitors for the treatment of cancer 薛定谔公司 2023-07-25 CN disclosed
EP-4211140-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER Schrödinger, Inc. (US) 2023-07-19 EP disclosed
US-20230101747-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. 2023-03-30 US disclosed
EP-4069369-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME Schrödinger, Inc. (US) 2022-10-12 EP disclosed
WO-2022055963-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. (US) 2022-03-17 WO disclosed
WO-2021113492-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. (US) 2021-06-10 WO disclosed
WO-2021113492-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME SCHRÖDINGER, INC. (US) 2021-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER CDC7, BUB1B, CDK7 COMT 4119/4885SMN1; SMN2 3929/4885ALDH1A1 3059/4885
US-20230101747-A1 CYCLIC COMPOUNDS AND METHODS OF USING SAME PLK1, DCK, CSNK1A1 COMT 4205/4885SMN1; SMN2 4423/4885ALDH1A1 2801/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.