SCHEMBL30002009

SCHEMBL30002009

O=Cc1c(F)c(F)cc2c1OCCO2

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
ACLY P53396 1/20 0.33
PKM P14618 8/20 0.32
PKLR P30613 6/20 0.32
ERN1 O75460 1/20 0.31
CTNNB1 P35222 1/20 0.31
WNT3A P56704 1/20 0.31
USP9X Q93008 1/20 0.31
PTGS2 P35354 2/20 0.31
TDP1 Q9NUW8 2/20 0.31
PTGS1 P23219 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892390 1.00 KDM4E (0.35) KDM4EACLYPKMPKLRERN1
SCHEMBL28581319 0.78 KDM4E (0.40) KDM4EACLYPKMPKLRERN1
SCHEMBL1058342 0.73 ALDH1A1 (0.43) KDM4EACLYERN1CTNNB1WNT3A
SCHEMBL18106671 0.70 ERN1 (0.36) PKMERN1TDP1
SCHEMBL909951 0.69 LMNA (0.42) PKMPKLRERN1TDP1ALDH1A1
SCHEMBL441131 0.69 CA1 (0.44) ERN1TDP1ALDH1A1MEN1KMT2A
SCHEMBL28892613 0.68
SCHEMBL28892511 0.68 CTNNB1 (0.31) CTNNB1WNT3A
SCHEMBL30002686 0.68 CTNNB1 (0.31) CTNNB1WNT3A
SCHEMBL30002413 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed