SCHEMBL30002067

SCHEMBL30002067

COc1cc(F)c(N)cc1OCc1c(F)ccc2scnc12

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.35
ERBB2 P04626 1/20 0.32
EPHA2 P29317 1/20 0.32
KDR P35968 1/20 0.32
PIK3CG P48736 1/20 0.32
GNRHR P30968 1/20 0.32
ALDH1A1 P00352 2/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TP53 P04637 1/20 0.30
PKM P14618 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892774 1.00 KIT (0.35) KITERBB2EPHA2KDRPIK3CG
SCHEMBL30002766 0.90 EPHA2 (0.37) KITERBB2EPHA2KDRNPC1
SCHEMBL28892550 0.90 EPHA2 (0.37) KITERBB2EPHA2KDRNPC1
SCHEMBL28892349 0.83 KIT (0.34) KITEPHA2KDRPIK3CGALDH1A1
SCHEMBL30002757 0.83 KIT (0.34) KITEPHA2KDRPIK3CGALDH1A1
SCHEMBL30003289 0.81 GAA (0.35) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL28892418 0.81 KIT (0.37) KITERBB2EPHA2KDRPIK3CG
SCHEMBL30003338 0.81 KIT (0.37) KITERBB2EPHA2KDRPIK3CG
SCHEMBL30002017 0.80 NPC1 (0.35) KITERBB2EPHA2KDRNPC1
SCHEMBL28892399 0.79 KIT (0.39) KITERBB2EPHA2KDRPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed