SCHEMBL30003289

SCHEMBL30003289

COc1cc(F)c([N+](=O)[O-])cc1OCc1c(F)ccc2scnc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.35
PKM P14618 1/20 0.35
ALDH1A1 P00352 8/20 0.34
LMNA P02545 3/20 0.34
CASP3 P42574 2/20 0.34
SENP8 Q96LD8 2/20 0.34
SENP7 Q9BQF6 2/20 0.34
SENP6 Q9GZR1 2/20 0.34
MEN1 O00255 5/20 0.34
KMT2A Q03164 5/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 4/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
PRKDC P78527 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CHEK1 O14757 2/20 0.34
MAPK1 P28482 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30002751 0.91 LMNA (0.35) GAAPKMALDH1A1LMNACASP3
SCHEMBL30002621 0.84 GAA (0.40) GAAPKMALDH1A1LMNACASP3
SCHEMBL28892761 0.84 GAA (0.40) GAAPKMALDH1A1LMNACASP3
SCHEMBL30002826 0.84 ALDH1A1 (0.37) GAAPKMALDH1A1LMNACASP3
SCHEMBL28892725 0.83 ALDH1A1 (0.36) GAAPKMALDH1A1LMNACASP3
SCHEMBL30002458 0.83 ALDH1A1 (0.36) GAAPKMALDH1A1LMNACASP3
SCHEMBL30002747 0.82 LMNA (0.34) GAAPKMALDH1A1LMNACASP3
SCHEMBL28892774 0.81 KIT (0.35) PKMALDH1A1MEN1KMT2ARAB9A
SCHEMBL30002067 0.81 KIT (0.35) PKMALDH1A1MEN1KMT2ARAB9A
SCHEMBL28892558 0.81 LMNA (0.38) GAAPKMALDH1A1LMNACASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed