SCHEMBL30002385

SCHEMBL30002385

COc1ccc(N2C(=O)c3ccccc3C2=O)c(F)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 1/20 0.68
NR1H3 Q13133 5/20 0.51
ESR1 P03372 2/20 0.51
NR1H2 P55055 2/20 0.50
ESR2 Q92731 1/20 0.49
ALDH1A1 P00352 3/20 0.45
HPGD P15428 2/20 0.45
KMT2A Q03164 2/20 0.45
CASP1 P29466 1/20 0.45
KDM4E B2RXH2 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP3A4 P08684 1/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GRM1 Q13255 1/20 0.44
GRM4 Q14833 1/20 0.44
ALOX15 P16050 1/20 0.44
GRM5 P41594 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3106326 1.00 SCN2A (0.68) SCN2ANR1H3ESR1NR1H2ESR2
SCHEMBL11808285 0.83 ESR1 (0.72) SCN2ANR1H3ESR1NR1H2ALDH1A1
SCHEMBL9216463 0.83 SCN2A (0.70) SCN2ANR1H3ESR1NR1H2ESR2
SCHEMBL9235862 0.81 SCN2A (0.68) SCN2ANR1H3ESR1NR1H2ALDH1A1
SCHEMBL6392226 0.79 SCN2A (0.66) SCN2ANR1H3ESR1NR1H2ALDH1A1
SCHEMBL6678239 0.79 ESR1 (0.53) SCN2ANR1H3ESR1NR1H2ESR2
SCHEMBL30273450 0.79 ESR1 (0.53) SCN2ANR1H3ESR1NR1H2ESR2
SCHEMBL10626656 0.78 ESR1 (0.56) SCN2AESR1ESR2KMT2ACASP1
SCHEMBL7729256 0.76 MEN1 (0.53) SCN2AESR1ESR2ALDH1A1KMT2A
SCHEMBL5924351 0.76 CYP3A4 (0.66) SCN2ANR1H3ESR1NR1H2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed