SCHEMBL30002609

SCHEMBL30002609

COc1cc(F)c(N)cc1OCc1cccc2sc(C)nc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 5/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
TSHR P16473 1/20 0.36
ALDH1A1 P00352 3/20 0.34
MPO P05164 1/20 0.34
PDE10A Q9Y233 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
PKM P14618 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
DHFR P00374 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892313 1.00 TDP1 (0.40) TDP1CYP3A4MAPTMEN1KMT2A
SCHEMBL28892521 0.83 GAA (0.39) MAPTMEN1KMT2AKDM4EGAA
SCHEMBL30002023 0.83 GAA (0.39) MAPTMEN1KMT2AKDM4EGAA
SCHEMBL30002757 0.82 KIT (0.34) TDP1CYP3A4MEN1KMT2AALDH1A1
SCHEMBL28892349 0.82 KIT (0.34) TDP1CYP3A4MEN1KMT2AALDH1A1
SCHEMBL30002421 0.80 MEN1 (0.47) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL28892709 0.79 KDM4E (0.39) KDM4EMPOPDE10ASMN1; SMN2CSF1R
SCHEMBL30002400 0.79 KDM4E (0.39) KDM4EMPOPDE10ASMN1; SMN2CSF1R
SCHEMBL28892336 0.78 SMN1; SMN2 (0.36) TDP1MAPTMEN1KMT2AKDM4E
SCHEMBL30002031 0.77 DHFR (0.38) TDP1MAPTMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed