SCHEMBL30002400

SCHEMBL30002400

COc1cc(F)c(N)cc1OCc1cccc2cc(C)cnc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
PSMD14 O00487 1/20 0.39
COPS5 Q92905 1/20 0.39
PDE10A Q9Y233 3/20 0.39
PARP1 P09874 1/20 0.38
CCR1 P32246 2/20 0.36
CCR5 P51681 2/20 0.36
CCR8 P51685 2/20 0.36
PIK3CD O00329 1/20 0.36
SLC40A1 Q9NP59 2/20 0.36
CSF1R P07333 1/20 0.36
TRPC6 Q9Y210 2/20 0.35
HPGDS O60760 1/20 0.35
MPO P05164 1/20 0.35
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892709 1.00 KDM4E (0.39) KDM4EPSMD14COPS5PDE10APARP1
SCHEMBL30002480 0.89 PDE10A (0.38) PDE10APIK3CDCSF1RHPGDSMPO
SCHEMBL30002421 0.83 MEN1 (0.47) KDM4EPDE10ASLC40A1CSF1R
SCHEMBL30002629 0.83 HTR1A (0.41) KDM4EPSMD14COPS5SMN1; SMN2
SCHEMBL30002661 0.81 MTNR1A (0.43) PDE10AMPO
SCHEMBL30002609 0.79 TDP1 (0.40) KDM4EPDE10ACSF1RMPOSMN1; SMN2
SCHEMBL28892336 0.79 SMN1; SMN2 (0.36) KDM4EPDE10ACSF1RMPOTP53
SCHEMBL28892313 0.79 TDP1 (0.40) KDM4EPDE10ACSF1RMPOSMN1; SMN2
SCHEMBL30002031 0.78 DHFR (0.38) CSF1RMPOSMN1; SMN2
SCHEMBL30002548 0.78 SCN1A (0.47) PDE10AMPOSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed