SCHEMBL30002665

SCHEMBL30002665

COc1cc(F)c(N)cc1OCc1ccc(Cl)c2ccncc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN8A Q9UQD0 1/20 0.37
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
KDR P35968 5/20 0.36
FLT1 P17948 2/20 0.36
EPHA2 P29317 4/20 0.36
ERBB2 P04626 2/20 0.36
EPHB4 P54760 2/20 0.36
KIT P10721 1/20 0.35
MGAT2 Q10469 1/20 0.35
G6PD P11413 1/20 0.34
GAA P10253 2/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PLK1 P53350 1/20 0.34
CSNK1A1 P48729 1/20 0.34
CSNK1D P48730 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892667 1.00 SCN1A (0.37) SCN1ASCN5ASCN8AIDO1TDO2
SCHEMBL30002637 0.90 KIT (0.37) SCN1ASCN5ASCN8AKDRFLT1
SCHEMBL28892213 0.90 KIT (0.37) SCN1ASCN5ASCN8AKDRFLT1
SCHEMBL30002084 0.85 KDR (0.37) IDO1TDO2KDRFLT1EPHA2
SCHEMBL28892434 0.85 KDR (0.37) IDO1TDO2KDRFLT1EPHA2
SCHEMBL28892367 0.83 KMT2A (0.41) SCN1ASCN5ASCN8AKDRFLT1
SCHEMBL30002548 0.81 SCN1A (0.47) SCN1ASCN5ASCN8AGAAMAPT
SCHEMBL28892526 0.81 SCN1A (0.47) SCN1ASCN5ASCN8AGAAMAPT
SCHEMBL30002702 0.79 KIT (0.37) IDO1TDO2KDRFLT1EPHA2
SCHEMBL28892670 0.79 KIT (0.37) IDO1TDO2KDRFLT1EPHA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed