SCHEMBL30002548

SCHEMBL30002548

COc1cc(F)c(N)cc1OCc1cccc2ccncc12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.47
SCN5A Q14524 1/20 0.47
SCN8A Q9UQD0 1/20 0.47
ADORA2A P29274 1/20 0.43
MAPT P10636 3/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
GRM2 Q14416 1/20 0.39
PARP15 Q460N3 1/20 0.38
PARP10 Q53GL7 1/20 0.38
PDE10A Q9Y233 5/20 0.38
MAOA P21397 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MPO P05164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892526 1.00 SCN1A (0.47) SCN1ASCN5ASCN8AADORA2AMAPT
SCHEMBL28892213 0.84 KIT (0.37) SCN1ASCN5ASCN8AMAPTGAA
SCHEMBL30002637 0.84 KIT (0.37) SCN1ASCN5ASCN8AMAPTGAA
SCHEMBL30002926 0.83 KIT (0.41)
SCHEMBL28892234 0.83 MAOA (0.39) MAPTGAASMN1; SMN2TDP1PDE10A
SCHEMBL30002556 0.83 MAOA (0.39) MAPTGAASMN1; SMN2TDP1PDE10A
SCHEMBL30002055 0.82 SCN1A (0.46) SCN1ASCN5ASCN8AADORA2AMAPT
SCHEMBL28893045 0.82 SCN1A (0.46) SCN1ASCN5ASCN8AADORA2AMAPT
SCHEMBL30002665 0.81 SCN1A (0.37) SCN1ASCN5ASCN8AMAPTGAA
SCHEMBL28892667 0.81 SCN1A (0.37) SCN1ASCN5ASCN8AMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed