SCHEMBL30002637

SCHEMBL30002637

COc1cc(F)c(N)cc1OCc1ccc(F)c2ccncc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.37
MGAT2 Q10469 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
FLT1 P17948 1/20 0.36
KDR P35968 1/20 0.36
RET P07949 1/20 0.35
KIF5B P33176 1/20 0.35
DGAT2 Q96PD7 3/20 0.34
MAOA P21397 2/20 0.34
PLK1 P53350 1/20 0.34
AURKA O14965 1/20 0.33
TTK P33981 1/20 0.33
AURKB Q96GD4 1/20 0.33
INCENP Q9NQS7 1/20 0.33
PDPK1 O15530 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892213 1.00 KIT (0.37) KITMGAT2SMN1; SMN2GAAMAPT
SCHEMBL30002665 0.90 SCN1A (0.37) KITMGAT2SMN1; SMN2GAAMAPT
SCHEMBL28892667 0.90 SCN1A (0.37) KITMGAT2SMN1; SMN2GAAMAPT
SCHEMBL28892526 0.84 SCN1A (0.47) SMN1; SMN2GAAMAPTTDP1MAOA
SCHEMBL30002548 0.84 SCN1A (0.47) SMN1; SMN2GAAMAPTTDP1MAOA
SCHEMBL28892670 0.84 KIT (0.37) KITSMN1; SMN2GAAMAPTTDP1
SCHEMBL30002702 0.84 KIT (0.37) KITSMN1; SMN2GAAMAPTTDP1
SCHEMBL28892812 0.81 CHEK1 (0.41) GAAMAPTTDP1RAB9AMEN1
SCHEMBL30002556 0.81 MAOA (0.39) KITSMN1; SMN2GAAMAPTTDP1
SCHEMBL28892234 0.81 MAOA (0.39) KITSMN1; SMN2GAAMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed