SCHEMBL30002819

SCHEMBL30002819

Fc1ccc2ccncc2c1CBr

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.38
DYRK1A Q13627 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.35
TNF P01375 2/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
MAPT P10636 3/20 0.33
MAPK10 P53779 3/20 0.33
HIPK2 Q9H2X6 1/20 0.33
IMPDH2 P12268 2/20 0.33
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
RAD52 P43351 1/20 0.32
P4HB P07237 1/20 0.32
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892447 1.00 CLK1 (0.38) CLK1DYRK1ALOXL2TNFHTR2A
SCHEMBL28892311 0.82 TNF (0.39) CLK1DYRK1ALOXL2TNFHTR2A
SCHEMBL30002436 0.79 KDM4E (0.37) LOXL2TNFMAPTHIPK2KDM4E
SCHEMBL28892698 0.79 KDM4E (0.37) LOXL2TNFMAPTHIPK2KDM4E
SCHEMBL30709993 0.76 IMPDH2 (0.43) CLK1DYRK1ALOXL2TNFHTR2A
SCHEMBL15058583 0.76 IMPDH2 (0.43) CLK1DYRK1ALOXL2TNFHTR2A
SCHEMBL28892536 0.75 LOXL2 (0.35) DYRK1ALOXL2KDM4EACHE
SCHEMBL30001957 0.75 LOXL2 (0.35) DYRK1ALOXL2KDM4EACHE
SCHEMBL22094381 0.75 CLK1 (0.43) CLK1DYRK1ALOXL2TNFHTR2A
SCHEMBL30308307 0.75 CLK1 (0.43) CLK1DYRK1ALOXL2TNFHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed