SCHEMBL30003152

SCHEMBL30003152

COc1cc(F)c(N)cc1OCc1c(F)cc(F)c2nccnc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.36
NSD2 O96028 1/20 0.35
CASP6 P55212 1/20 0.35
G6PD P11413 1/20 0.35
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HTR2A P28223 3/20 0.31
ERBB2 P04626 1/20 0.31
EPHA2 P29317 1/20 0.31
KDR P35968 1/20 0.31
CCNB2 O95067 1/20 0.30
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
GSK3A P49840 1/20 0.30
GSK3B P49841 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30
CCNB3 Q8WWL7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892632 1.00 KIT (0.36) KITNSD2CASP6G6PDGAA
SCHEMBL28959473 0.84 NSD2 (0.47) KITNSD2CASP6G6PDGAA
SCHEMBL30002712 0.84 NSD2 (0.47) KITNSD2CASP6G6PDGAA
SCHEMBL28892399 0.84 KIT (0.39) KITNSD2CASP6G6PDGAA
SCHEMBL30003339 0.84 KIT (0.39) KITNSD2CASP6G6PDGAA
SCHEMBL28892170 0.81 KIT (0.36) KITNSD2CASP6G6PDGAA
SCHEMBL30002605 0.81 KIT (0.36) KITNSD2CASP6G6PDGAA
SCHEMBL28892537 0.79 NSD2 (0.41) NSD2CASP6G6PDGAAMAPT
SCHEMBL28892693 0.79 KMT2A (0.39) GAAMAPT
SCHEMBL30003250 0.79 NSD2 (0.41) NSD2CASP6G6PDGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed