SCHEMBL28892170

SCHEMBL28892170

COc1cc(F)c(N)cc1OCc1c(F)c(F)cc2nccnc12

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.36
NSD2 O96028 1/20 0.33
CASP6 P55212 1/20 0.33
G6PD P11413 1/20 0.33
PDPK1 O15530 1/20 0.32
MET P08581 1/20 0.32
ERBB2 P04626 1/20 0.31
EPHA2 P29317 1/20 0.31
KDR P35968 1/20 0.31
EHMT2 Q96KQ7 1/20 0.31
EHMT1 Q9H9B1 1/20 0.31
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
CSF1R P07333 1/20 0.30
ENPP1 P22413 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30002605 1.00 KIT (0.36) KITNSD2CASP6G6PDPDPK1
SCHEMBL28892399 0.85 KIT (0.39) KITNSD2CASP6G6PDERBB2
SCHEMBL30003339 0.85 KIT (0.39) KITNSD2CASP6G6PDERBB2
SCHEMBL30002638 0.82 NSD2 (0.41) KITNSD2CASP6G6PDGAA
SCHEMBL28892621 0.82 NSD2 (0.41) KITNSD2CASP6G6PDGAA
SCHEMBL30003152 0.81 KIT (0.36) KITNSD2CASP6G6PDERBB2
SCHEMBL28892632 0.81 KIT (0.36) KITNSD2CASP6G6PDERBB2
SCHEMBL28892567 0.81 KMT2A (0.41) GAAMAPT
SCHEMBL30002050 0.81 KMT2A (0.41) GAAMAPT
SCHEMBL4301135 0.77 GNRHR (0.43) KITGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed