SCHEMBL30003339

SCHEMBL30003339

COc1cc(F)c(N)cc1OCc1c(F)ccc2nccnc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
KDR P35968 4/20 0.35
ERBB2 P04626 1/20 0.35
EPHA2 P29317 1/20 0.35
NSD2 O96028 1/20 0.35
CASP6 P55212 1/20 0.35
G6PD P11413 1/20 0.35
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
EHMT1 Q9H9B1 1/20 0.33
FLT1 P17948 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892399 1.00 KIT (0.39) KITMEN1KMT2AKDRERBB2
SCHEMBL30002605 0.85 KIT (0.36) KITKDRERBB2EPHA2NSD2
SCHEMBL28892170 0.85 KIT (0.36) KITKDRERBB2EPHA2NSD2
SCHEMBL30003152 0.84 KIT (0.36) KITKDRERBB2EPHA2NSD2
SCHEMBL28892632 0.84 KIT (0.36) KITKDRERBB2EPHA2NSD2
SCHEMBL28892537 0.83 NSD2 (0.41) MEN1KMT2ANSD2CASP6G6PD
SCHEMBL30003250 0.83 NSD2 (0.41) MEN1KMT2ANSD2CASP6G6PD
SCHEMBL30002031 0.82 DHFR (0.38) KITMEN1KMT2AKDREPHA2
SCHEMBL30003416 0.81 KMT2A (0.50) MEN1KMT2AGAAMAPTPDGFRB
SCHEMBL28892412 0.81 KMT2A (0.50) MEN1KMT2AGAAMAPTPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed