SCHEMBL30004753

SCHEMBL30004753

NC(=O)c1cccc(C2CO2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 1.00
TSHR P16473 3/20 0.45
KDM1A O60341 2/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
OPRM1 P35372 4/20 0.42
OPRD1 P41143 4/20 0.42
POLB P06746 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C19 P33261 1/20 0.42
RECQL P46063 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
PARP10 Q53GL7 2/20 0.41
TNKS O95271 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4274420 0.84 PARP1 (0.72) PARP1TSHRHSD17B10
SCHEMBL1499340 0.82 PARP1 (0.70) PARP1TSHRMAPTTDP1
SCHEMBL6697278 0.81 PARP1 (0.68) PARP1TSHRKDM1AMAOAMAOB
Aniline SCHEMBL28655458 0.79 PARP1 (0.65) PARP1TSHRKDM1AMAOAHSD17B10
SCHEMBL1036815 0.78 PARP1 (0.64) PARP1OPRM1OPRD1HRH3PARP14
Hydrochloric Acid SCHEMBL30520457 0.78 PARP1 (0.62) PARP1
Phenol SCHEMBL28650467 0.77 PARP1 (0.62) PARP1TSHR
SCHEMBL21974861 0.76 TSHR (0.67) PARP1TSHRCYP3A4CYP2C19
SCHEMBL46283 0.76 TSHR (0.67) PARP1TSHRCYP3A4CYP2C19
SCHEMBL29503161 0.75 KMO (0.65) PARP1OPRM1OPRD1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022220725-A1 LPXH INHIBITORS AS ANTI-INFECTIVE AGENTS ZAMARATSKI EDOUARD (SE) 2022-10-20 WO disclosed