SCHEMBL30005432

SCHEMBL30005432

Nc1cc(F)cc(OC(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.40
BACE1 P56817 3/20 0.35
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19950199 1.00 APP (0.40) APPBACE1ALDH1A1MAPT
SCHEMBL1494673 0.77 ALOX15 (0.32) APPALDH1A1MAPT
SCHEMBL22081760 0.77 CYP3A4 (0.48) APPALDH1A1MAPT
SCHEMBL30004351 0.77 CYP3A4 (0.48) APPALDH1A1MAPT
SCHEMBL30345392 0.77 ALOX15 (0.32) APPALDH1A1MAPT
SCHEMBL24803973 0.77 ALDH1A1 (0.31) APPALDH1A1MAPT
SCHEMBL8999877 0.77 MEN1 (0.43) ALDH1A1MAPT
SCHEMBL1100004 0.75 MEN1 (0.47) ALDH1A1MAPT
SCHEMBL3157193 0.74 ALOX15 (0.32) APP
SCHEMBL17203920 0.74 APP (0.34) APPBACE1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4323350-A1 ISOINDOLINONE COMPOUNDS Monte Rosa Therapeutics AG (CH) 2024-02-21 EP disclosed
CN-117242060-A Isoindolinone compounds 蒙特罗萨医疗公司 2023-12-15 CN disclosed
WO-2023069731-A1 COMPOUNDS THAT MEDIATE PROTEIN DEGRADATION AND METHODS OF USE THEREOF MONTE ROSA THERAPEUTICS, INC. (US) 2023-04-27 WO disclosed
CN-115819417-A Pyrazolopyridine derivatives as HPK1 modulators and their use for the treatment of cancer 因赛特公司 2023-03-21 CN disclosed
CN-109923114-B Pyrazolopyridine derivatives as HPK1 modulators and their use for the treatment of cancer 因赛特公司 2022-11-01 CN disclosed
WO-2022219407-A1 ISOINDOLINONE COMPOUNDS MONTE ROSA THERAPEUTICS AG (CH) 2022-10-20 WO disclosed