SCHEMBL30006316

SCHEMBL30006316

C[C@@H](N)c1cc(N)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 9/20 0.43
KRAS P01116 6/20 0.43
TACR1 P25103 4/20 0.43
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
PDE2A O00408 1/20 0.40
PNMT P11086 1/20 0.40
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
NR2E1 Q9Y466 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
CACNA1F O60840 1/20 0.35
CACNA1D Q01668 1/20 0.35
CACNA1S Q13698 1/20 0.35
CACNA1C Q13936 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20327218 1.00 SOS1 (0.43) SOS1KRASTACR1TSHRMAPK1
SCHEMBL12587301 1.00 SOS1 (0.43) SOS1KRASTACR1TSHRMAPK1
Hydrochloric Acid SCHEMBL23326533 0.98 SOS1 (0.42) SOS1KRASTACR1TSHRMAPK1
Hydrochloric Acid SCHEMBL29564024 0.98 SOS1 (0.42) SOS1KRASTACR1TSHRMAPK1
Hydrochloric Acid SCHEMBL23326532 0.98 SOS1 (0.42) SOS1KRASTACR1TSHRMAPK1
Hydrochloric Acid SCHEMBL29663260 0.98 SOS1 (0.42) SOS1KRASTACR1TSHRMAPK1
SCHEMBL336049 0.87 TACR1 (0.51) TACR1PDE2APNMTIDO1TDO2
SCHEMBL7939177 0.87 TACR1 (0.51) TACR1PDE2APNMTIDO1TDO2
SCHEMBL1728680 0.87 TACR1 (0.51) TACR1PDE2APNMTIDO1TDO2
SCHEMBL6917133 0.87 TACR1 (0.51) TACR1PDE2APNMTIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119039234-B Pyridazine amide compound and preparation method and application thereof 中国药科大学 2026-05-15 CN disclosed
CN-119431234-A Benzyl amine formyl compound and preparation method and application thereof 中国药科大学 2025-02-14 CN disclosed
CN-119039234-A Pyridazine amide compound and preparation method and application thereof 中国药科大学 2024-11-29 CN disclosed
EP-4322962-A1 PHOSPHORUS DERIVATIVES AS NOVEL SOS1 INHIBITORS Bayer Aktiengesellschaft (DE) 2024-02-21 EP disclosed
WO-2022219035-A1 PHOSPHORUS DERIVATIVES AS NOVEL SOS1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2022-10-20 WO disclosed