SCHEMBL30006948

SCHEMBL30006948

C=C(c1nc(-c2ccc(F)cc2)c(F)c(C(C)(C)O)c1F)C1CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
CFTR P13569 3/20 0.33
NR3C1 P04150 6/20 0.31
TNIK Q9UKE5 1/20 0.31
SLC34A1 Q06495 1/20 0.31
PGR P06401 1/20 0.31
HRH2 P25021 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
ACHE P22303 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
BRAF P15056 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
TGFBR1 P36897 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958662 1.00 ADORA2A (0.33) ADORA2AADORA2BADORA1CFTRNR3C1
SCHEMBL30007397 0.90 SLC34A1 (0.34) ADORA2AADORA2BADORA1CFTRNR3C1
SCHEMBL25686856 0.90 SLC34A1 (0.34) ADORA2AADORA2BADORA1CFTRNR3C1
SCHEMBL25423458 0.83 CFTR (0.37) CFTRBRAFMEN1KMT2A
SCHEMBL26727261 0.76 CFTR (0.34) ADORA2AADORA2BADORA1CFTRTNIK
SCHEMBL30007279 0.74 SLC34A1 (0.35) ADORA2AADORA2BADORA1SLC34A1BRAF
SCHEMBL23958637 0.74 SLC34A1 (0.35) ADORA2AADORA2BADORA1SLC34A1BRAF
SCHEMBL28960596 0.73 CFTR (0.32) CFTRTNIKTGFBR1MEN1KMT2A
SCHEMBL23958949 0.72 CFTR (0.35) ADORA2AADORA1CFTRSLC34A1BRAF
SCHEMBL23958787 0.71 SLC34A1 (0.33) CFTRNR3C1SLC34A1HRH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed