SCHEMBL30007189

SCHEMBL30007189

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)cc(-c3ccc(F)c(F)c3)n2)C2CC2)cc2cc(C)nnc12

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.33
MAPK14 Q16539 1/20 0.33
GABRA5 P31644 2/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
CNR1 P21554 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
CTSA P10619 1/20 0.30
MEN1 O00255 3/20 0.30
KMT2A Q03164 3/20 0.30
MAPT P10636 2/20 0.30
RAB9A P51151 1/20 0.30
ACACB O00763 1/20 0.30
ACACA Q13085 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25234972 1.00 CYP2C9 (0.33) CYP2C9MAPK14GABRA5ALDH1A1POLB
SCHEMBL25687466 0.93 SCN9A (0.36) CYP2C9MAPK14ROCK2ROCK1ACACB
SCHEMBL25687467 0.93 SCN9A (0.36) CYP2C9MAPK14ROCK2ROCK1ACACB
SCHEMBL30007220 0.93 SCN9A (0.36) CYP2C9MAPK14ROCK2ROCK1ACACB
SCHEMBL28909130 0.93 SCN9A (0.36) CYP2C9MAPK14ROCK2ROCK1ACACB
SCHEMBL30007118 0.87 CTSA (0.35) CYP2C9MAPK14GABRA5ROCK2ROCK1
SCHEMBL23958892 0.87 CTSA (0.35) CYP2C9MAPK14GABRA5ROCK2ROCK1
SCHEMBL25687368 0.87 CTSA (0.35) CYP2C9MAPK14GABRA5ROCK2ROCK1
SCHEMBL30007246 0.81 CNR1 (0.37) CYP2C9MAPK14GABRA5ALDH1A1ROCK2
SCHEMBL28909201 0.81 CNR1 (0.37) CYP2C9MAPK14GABRA5ALDH1A1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed