SCHEMBL30007248

SCHEMBL30007248

CCN(CC)c1ccc(CNC(=O)c2n[nH]c3ncc(-c4ccc(S(=O)(=O)C(C)C)cc4)cc23)cc1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.40
DYRK1A Q13627 8/20 0.38
CLK1 P49759 1/20 0.38
WNT1 P04628 3/20 0.37
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NAMPT P43490 5/20 0.36
GSK3B P49841 1/20 0.35
ROCK2 O75116 1/20 0.35
CNR2 P34972 1/20 0.35
MAP4K1 Q92918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30007830 0.88 DYRK1A (0.45) ATRDYRK1AWNT1NAMPTGSK3B
SCHEMBL30008206 0.85 CLK1 (0.43) ATRDYRK1ACLK1NAMPTGSK3B
SCHEMBL30007739 0.82 NAMPT (0.43) ATRNAMPT
SCHEMBL30007902 0.77 GSK3A (0.46) ATRDYRK1AGSK3B
SCHEMBL30007683 0.75 CYP2C9 (0.48) DYRK1ACLK1NAMPTGSK3B
SCHEMBL30007677 0.71 AXL (0.50) NAMPT
SCHEMBL29253947 0.69 GSK3A (0.48) ATRDYRK1AGSK3B
SCHEMBL30912733 0.69 GSK3B (0.46) DYRK1AGSK3B
SCHEMBL30912725 0.69 GSK3B (0.46) DYRK1AGSK3B
SCHEMBL29253944 0.69 GSK3B (0.46) DYRK1AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO claimed
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO disclosed